SCHEMBL1275918

SCHEMBL1275918

COc1cccc2c1C/C(=C/CCN1CCC(n3c(=O)[nH]c4ccccc43)CC1)c1cccnc1O2

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.46
DRD3 P35462 2/20 0.46
DRD4 P21917 1/20 0.46
CHRM1 P11229 5/20 0.45
KCNH2 Q12809 3/20 0.45
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
PLD2 O14939 2/20 0.44
PLD1 Q13393 2/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
OPRM1 P35372 8/20 0.43
OPRL1 P41146 6/20 0.43
HTR1A P08908 1/20 0.43
CHRM5 P08912 1/20 0.43
HTR2A P28223 1/20 0.43
OPRD1 P41143 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL652632 1.00 DRD2 (0.46) DRD2DRD3DRD4CHRM1KCNH2
SCHEMBL652357 0.91 DRD2 (0.47) DRD2DRD3DRD4CHRM1KCNH2
SCHEMBL656124 0.88 SIGMAR1 (0.42) OPRM1OPRL1HTR1A
SCHEMBL653247 0.82 ABCB1 (0.48) DRD4CHRM1KCNH2HTR1ACHRM5
SCHEMBL653245 0.82 ABCB1 (0.48) DRD4CHRM1KCNH2HTR1ACHRM5
SCHEMBL652340 0.82 SIGMAR1 (0.45) HTR1A
SCHEMBL652338 0.82 SIGMAR1 (0.45) HTR1A
SCHEMBL653232 0.81 SIGMAR1 (0.46) DRD2DRD3DRD4KCNH2HTR1A
SCHEMBL653234 0.81 SIGMAR1 (0.46) DRD2DRD3DRD4KCNH2HTR1A
SCHEMBL655814 0.80 SLC6A4 (0.42) CYP2D6ADRA1DHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2286811-A1 Chemokine receptor antagonists and methods of use thereof Millennium Pharmaceuticals, Inc. (US) 2011-02-23 EP disclosed