SCHEMBL12779481

SCHEMBL12779481

CCn1nc(C(=O)N(Cc2ccncc2)CN(C)C)c2ccc(-c3cn[nH]c3)cc21

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 15/20 0.43
ROCK2 O75116 14/20 0.43
PRKACA P17612 2/20 0.43
PRKACG P22612 2/20 0.43
PRKACB P22694 2/20 0.43
METAP2 P50579 1/20 0.38
CDC42BPA Q5VT25 2/20 0.36
MAPK10 P53779 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12780552 0.86 ROCK2 (0.61) ROCK1ROCK2PRKACAPRKACGPRKACB
SCHEMBL12779480 0.83 ROCK2 (0.54) ROCK1ROCK2PRKACAPRKACGPRKACB
SCHEMBL12779506 0.80 ROCK2 (0.45) ROCK1ROCK2PRKACAPRKACGPRKACB
SCHEMBL12779550 0.78 ROCK2 (0.71) ROCK1ROCK2PRKACAPRKACGPRKACB
SCHEMBL12779294 0.78 ROCK2 (0.48) ROCK1ROCK2PRKACAPRKACGPRKACB
SCHEMBL12779442 0.76 ROCK1 (0.57) ROCK1ROCK2PRKACAPRKACGPRKACB
SCHEMBL12779510 0.75 ROCK2 (0.41) ROCK1ROCK2PRKACAPRKACGPRKACB
SCHEMBL1648217 0.69 ROCK2 (0.67) ROCK1ROCK2PRKACAPRKACGPRKACB
SCHEMBL12779448 0.64 ROCK2 (0.53) ROCK1ROCK2PRKACAPRKACGPRKACB
SCHEMBL1647834 0.62 PRKACA (0.77) ROCK1ROCK2PRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed