SCHEMBL12780552

SCHEMBL12780552

CCn1nc(C(=O)N(Cc2cccc(OC)c2)CN(C)C)c2ccc(-c3cn[nH]c3)cc21

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 17/20 0.61
ROCK1 Q13464 16/20 0.61
PRKACA P17612 2/20 0.60
PRKACG P22612 2/20 0.60
PRKACB P22694 2/20 0.60
CDC42BPA Q5VT25 4/20 0.53
CYP2C9 P11712 2/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
MAPK10 P53779 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12779550 0.93 ROCK2 (0.71) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779442 0.90 ROCK1 (0.57) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779481 0.86 ROCK1 (0.43) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1648217 0.83 ROCK2 (0.67) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779480 0.80 ROCK2 (0.54) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779448 0.79 ROCK2 (0.53) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779506 0.77 ROCK2 (0.45) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1647243 0.76 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1647834 0.76 PRKACA (0.77) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1648903 0.75 PRKACA (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed