SCHEMBL12779552

SCHEMBL12779552

COc1cccc(CN(C)C(=O)c2cc3ccc(-c4ccncc4)cc3[nH]2)c1

nearest known ligand 0.77

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 14/20 0.77
ROCK1 Q13464 14/20 0.77
RXFP1 Q9HBX9 2/20 0.66
MEN1 O00255 1/20 0.66
KMT2A Q03164 1/20 0.66
HSD17B2 P37059 2/20 0.57
PRKACA P17612 1/20 0.52
PRKACG P22612 1/20 0.52
PRKACB P22694 1/20 0.52
ABHD6 Q9BV23 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1649561 0.87 ROCK2 (1.00) ROCK2ROCK1RXFP1MEN1KMT2A
SCHEMBL12779204 0.87 ROCK2 (0.79) ROCK2ROCK1RXFP1MEN1KMT2A
SCHEMBL12779549 0.82 ROCK2 (1.00) ROCK2ROCK1MEN1KMT2APRKACA
SCHEMBL1649557 0.80 ROCK1 (0.76) ROCK2ROCK1HSD17B2PRKACAABHD6
SCHEMBL12779736 0.76 ROCK2 (0.80) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1647585 0.75 ROCK1 (0.78) ROCK2ROCK1HSD17B2ABHD6
SCHEMBL1647157 0.75 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779734 0.74 ROCK2 (0.79) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12495934 0.73 HSD17B2 (1.00) ROCK2ROCK1MEN1KMT2AHSD17B2
SCHEMBL1648507 0.73 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed