SCHEMBL1649561

SCHEMBL1649561

COc1cccc(CN(C)C(=O)c2cc3ccc(-c4cn[nH]c4)cc3[nH]2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 17/20 1.00
ROCK1 Q13464 13/20 1.00
PRKACA P17612 3/20 0.70
PRKACG P22612 3/20 0.70
PRKACB P22694 3/20 0.70
MEN1 O00255 1/20 0.64
KMT2A Q03164 1/20 0.64
RXFP1 Q9HBX9 1/20 0.64
CYP2C9 P11712 1/20 0.61
CDC42BPA Q5VT25 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12779736 0.89 ROCK2 (0.80) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1647157 0.87 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779734 0.87 ROCK2 (0.79) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779552 0.87 ROCK2 (0.77) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1648507 0.86 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1647875 0.83 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL12779554 0.82 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1647880 0.82 ROCK1 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1648742 0.81 ROCK2 (1.00) ROCK2ROCK1PRKACAPRKACGPRKACB
SCHEMBL1648748 0.81 ROCK2 (0.83) ROCK2ROCK1PRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed
WO-2011050245-A1 BICYCLIC HETEROARYLS AS KINASE INHIBITORS FENG YANGBO (US) 2011-04-28 WO disclosed