SCHEMBL12801536

SCHEMBL12801536

COc1cc(Nc2nccc(-c3ccc(OC4CCN(C(C)=O)CC4)c(N)c3)n2)cc(OC)c1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ZAP70 P43403 13/20 0.52
PRKD3 O94806 4/20 0.51
PRKCG P05129 4/20 0.51
PRKCB P05771 4/20 0.51
LCK P06239 4/20 0.51
PRKCA P17252 4/20 0.51
PRKCH P24723 4/20 0.51
PRKCI P41743 4/20 0.51
PRKCE Q02156 4/20 0.51
PRKCQ Q04759 4/20 0.51
PRKCZ Q05513 4/20 0.51
PRKCD Q05655 4/20 0.51
PRKD1 Q15139 4/20 0.51
EGFR P00533 3/20 0.51
JAK2 O60674 2/20 0.51
CDK2 P24941 2/20 0.51
PIK3CA P42336 1/20 0.51
PIK3CB P42338 1/20 0.51
PIK3CG P48736 1/20 0.51
PTK2B Q14289 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1667770 0.88 TBK1 (0.56) ZAP70JAK2
SCHEMBL12801104 0.83 JAK2 (0.47) ZAP70PRKD3PRKCGPRKCBLCK
SCHEMBL12800915 0.83 JAK2 (0.62) JAK2
SCHEMBL12801368 0.83 GSK3B (0.43) ZAP70JAK2CDK2IKBKBIGF1R
SCHEMBL12522369 0.82 SYK (0.40) EGFRJAK2CDK2IKBKBCHUK
SCHEMBL12801107 0.80 TBK1 (0.47) JAK2CDK2PIK3CGIKBKBCHUK
SCHEMBL1667112 0.80 TBK1 (0.53) JAK2
SCHEMBL12522198 0.79 TBK1 (0.52) JAK2SYK
SCHEMBL12521964 0.79 CCNC (0.47) ZAP70JAK2CDK2IKBKBIGF1R
SCHEMBL12801550 0.79 JAK2 (0.60) JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed