SCHEMBL12801550

SCHEMBL12801550

CC(=O)N1CCC(Oc2ccc(-c3ccnc(Nc4ccc(N5CCOCC5)cc4)n3)cc2N)C1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 19/20 0.60
JAK3 P52333 11/20 0.56
TBK1 Q9UHD2 2/20 0.53
JAK1 P23458 4/20 0.53
TYK2 P29597 3/20 0.53
HDAC3 O15379 1/20 0.52
NCOR1 O75376 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12800915 0.95 JAK2 (0.62) JAK2JAK3TBK1JAK1TYK2
SCHEMBL12800908 0.95 JAK2 (0.63) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12801569 0.92 JAK2 (0.57) JAK2JAK3TBK1JAK1TYK2
SCHEMBL12801563 0.91 JAK2 (0.57) JAK2JAK3TBK1JAK1TYK2
SCHEMBL12801254 0.91 JAK2 (0.57) JAK2JAK3TBK1JAK1TYK2
SCHEMBL12801176 0.91 JAK2 (0.64) JAK2JAK3TBK1JAK1TYK2
SCHEMBL12801574 0.90 JAK2 (0.55) JAK2JAK3TBK1JAK1TYK2
SCHEMBL12274829 0.89 TBK1 (0.67) JAK2TBK1
SCHEMBL12801257 0.89 JAK2 (0.59) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12801555 0.89 JAK2 (0.59) JAK2JAK3JAK1TYK2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed