SCHEMBL12801569

SCHEMBL12801569

Nc1cc(-c2ccnc(Nc3ccc(N4CCOCC4)cc3)n2)ccc1OC1CCN(C(=O)C2CC2)C1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 18/20 0.57
JAK3 P52333 9/20 0.53
JAK1 P23458 4/20 0.52
TYK2 P29597 4/20 0.52
TBK1 Q9UHD2 3/20 0.52
HDAC3 O15379 1/20 0.51
NCOR1 O75376 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
PDGFRB P09619 2/20 0.50
FLT3 P36888 2/20 0.50
IKBKB O14920 1/20 0.50
KIT P10721 1/20 0.50
PDGFRA P16234 1/20 0.50
FLT1 P17948 1/20 0.50
RPS6KB1 P23443 1/20 0.50
FLT4 P35916 1/20 0.50
KDR P35968 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801550 0.92 JAK2 (0.60) JAK2JAK3JAK1TYK2TBK1
SCHEMBL12801176 0.90 JAK2 (0.64) JAK2JAK3JAK1TYK2TBK1
SCHEMBL12801563 0.89 JAK2 (0.57) JAK2JAK3JAK1TYK2TBK1
SCHEMBL12801574 0.89 JAK2 (0.55) JAK2JAK3JAK1TYK2TBK1
SCHEMBL12801254 0.89 JAK2 (0.57) JAK2JAK3JAK1TYK2TBK1
SCHEMBL12522351 0.89 TBK1 (0.66) JAK2TBK1IKBKE
SCHEMBL12800915 0.89 JAK2 (0.62) JAK2JAK3JAK1TYK2TBK1
SCHEMBL12801555 0.88 JAK2 (0.59) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12800908 0.88 JAK2 (0.63) JAK2JAK3JAK1TYK2HDAC3
SCHEMBL12800922 0.87 JAK2 (0.58) JAK2JAK3JAK1TYK2TBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed