SCHEMBL12801596

SCHEMBL12801596

COc1ccc(Nc2nc(-c3cccc(N)c3)c3ccccc3n2)cc1OC

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.58
LMNA P02545 1/20 0.58
MAPK1 P28482 1/20 0.58
ABCG2 Q9UNQ0 14/20 0.57
ABCB1 P08183 9/20 0.57
ABCC1 P33527 4/20 0.57
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51
TP53 P04637 1/20 0.48
FLT3 P36888 1/20 0.48
CD63 P08962 1/20 0.48
SYK P43405 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801627 0.88 MAPT (0.56) MAPTLMNAMAPK1ABCG2ABCB1
SCHEMBL1667296 0.84 ABCG2 (0.60) MAPTLMNAMAPK1ABCG2ABCB1
SCHEMBL12275273 0.81 MAPT (0.53) MAPTLMNAMAPK1ABCG2ABCB1
SCHEMBL12274278 0.80 MAPT (0.60) MAPTLMNAMAPK1ABCG2ABCB1
SCHEMBL12801657 0.79 SYK (0.51) MEN1KMT2AFLT3CD63SYK
SCHEMBL12801284 0.78 PAK1 (0.53) MEN1KMT2AFLT3CD63SYK
SCHEMBL8899168 0.78 ABCG2 (0.72) MAPTLMNAABCG2ABCB1ABCC1
Hydrochloric Acid SCHEMBL8907536 0.77 ABCG2 (0.70) MAPTLMNAABCG2ABCB1ABCC1
SCHEMBL12801614 0.76 SYK (0.55) MAPTABCG2ABCB1ABCC1MEN1
SCHEMBL369450 0.75 PDE4A (0.59) MAPTABCG2MEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed