SCHEMBL12801657

SCHEMBL12801657

COc1ccc(Nc2ncc(C)c(-c3cccc(N)c3)n2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.51
CD63 P08962 1/20 0.51
MAPK8 P45983 1/20 0.50
MAPK9 P45984 1/20 0.50
PLK1 P53350 3/20 0.49
BRD4 O60885 1/20 0.49
KDR P35968 3/20 0.48
CDK5 Q00535 2/20 0.48
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48
CDK5R1 Q15078 1/20 0.48
EGFR P00533 1/20 0.45
ITK Q08881 1/20 0.45
FLT3 P36888 2/20 0.44
JAK2 O60674 2/20 0.43
AURKA O14965 1/20 0.43
KIT P10721 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801284 0.88 PAK1 (0.53) SYKCD63MAPK8MAPK9PLK1
SCHEMBL12274826 0.84 FLT3 (0.52) SYKPLK1KDRFLT3KIT
SCHEMBL12801596 0.79 MAPT (0.58) SYKCD63MEN1KMT2AFLT3
SCHEMBL17573404 0.78 KDR (0.49) SYKPLK1BRD4KDRCDK5
SCHEMBL8089927 0.77 SYK (0.54) SYKKDRCDK5EGFRJAK2
SCHEMBL12801614 0.77 SYK (0.55) SYKCD63PLK1CDK5MEN1
SCHEMBL14254047 0.74 ITK (0.53) SYKMAPK8MAPK9PLK1KDR
SCHEMBL12999380 0.74 JAK2 (0.52) MAPK8MAPK9PLK1BRD4KDR
SCHEMBL13169823 0.73 BRD4 (0.49) MAPK8MAPK9PLK1BRD4KDR
SCHEMBL4560068 0.73 JAK1 (0.58) BRD4KDRJAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed