SCHEMBL12822014

SCHEMBL12822014

Cc1c(C(N)=O)cccc1-n1cccc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
LMNA P02545 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
GAA P10253 2/20 0.46
CYP2C19 P33261 3/20 0.41
CYP2C9 P11712 2/20 0.41
NPC1 O15118 1/20 0.41
PARP1 P09874 2/20 0.40
POLB P06746 1/20 0.40
CYP1A2 P05177 2/20 0.39
MYC P01106 1/20 0.39
KDM4E B2RXH2 3/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11173849 0.84 MYC (0.51) ALDH1A1LMNAL3MBTL1CYP2C19CYP2C9
SCHEMBL5319528 0.81 IDO1 (0.47) ALDH1A1LMNAGAACYP2C19CYP2C9
SCHEMBL607557 0.81 ALDH1A1 (0.65) ALDH1A1LMNAL3MBTL1GAACYP2C19
SCHEMBL5789460 0.79 ALDH1A1 (0.49) ALDH1A1LMNAL3MBTL1GAACYP2C19
SCHEMBL5785069 0.78 ALDH1A1 (0.49) ALDH1A1LMNAL3MBTL1GAACYP2C19
SCHEMBL39964 0.78 KDM4E (0.52) ALDH1A1GAAPARP1KDM4EMAPT
Hydrochloric Acid SCHEMBL4562961 0.76 PARP1 (0.50) ALDH1A1GAAPARP1KDM4EMAPT
SCHEMBL28793930 0.76 NPC1 (0.63) ALDH1A1LMNAL3MBTL1GAANPC1
SCHEMBL27765492 0.76 NPC1 (0.44) ALDH1A1LMNAGAANPC1PARP1
SCHEMBL3684197 0.75 ALDH1A1 (0.45) ALDH1A1LMNAL3MBTL1GAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2691375-A1 SUBSTITUTED BENZIMIDAZOLES Bayer Intellectual Property GmbH (DE) 2014-02-05 EP claimed
WO-2012130905-A1 SUBSTITUTED BENZIMIDAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-10-04 WO claimed