SCHEMBL5789460

SCHEMBL5789460

NC(=O)c1cccc(-n2cccc2)c1F

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
LMNA P02545 4/20 0.48
GAA P10253 3/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPC1 O15118 1/20 0.41
KDM4E B2RXH2 3/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KMT2A Q03164 2/20 0.38
CES2 O00748 1/20 0.37
BCHE P06276 1/20 0.37
CES1 P23141 1/20 0.37
GPR52 Q9Y2T5 1/20 0.36
METAP2 P50579 1/20 0.36
OPRM1 P35372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29517255 0.84 LMNA (0.49) ALDH1A1LMNAGAAL3MBTL1CYP2C9
SCHEMBL607557 0.81 ALDH1A1 (0.65) ALDH1A1LMNAGAAL3MBTL1CYP2C9
SCHEMBL12822014 0.79 ALDH1A1 (0.49) ALDH1A1LMNAGAAL3MBTL1CYP2C9
SCHEMBL27214503 0.78 ALDH1A1 (0.52) ALDH1A1GAAKDM4EMAPTHPGD
SCHEMBL3684197 0.75 ALDH1A1 (0.45) ALDH1A1LMNAGAAL3MBTL1NPC1
SCHEMBL5785069 0.75 ALDH1A1 (0.49) ALDH1A1LMNAGAAL3MBTL1CYP2C9
SCHEMBL5784881 0.74 PARP1 (0.42) ALDH1A1LMNAGAAL3MBTL1NPC1
SCHEMBL5789102 0.73 POLB (0.44) ALDH1A1LMNAGAAL3MBTL1CYP2C9
SCHEMBL4096686 0.73 MAPT (0.44) ALDH1A1GAAL3MBTL1NPC1KDM4E
SCHEMBL29528396 0.72 CES2 (0.68) ALDH1A1GAANPC1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646610-A1 TETRAHYDROCARBAZOLE DERIVATIVES AND THEIR PHARMACEUTICAL USE SmithKline Beecham Corporation (US) 2006-04-19 EP disclosed
WO-2005005386-A1 TETRAHYDROCARBAZOLE DERIVATIVES AND THEIR PHARMACEUTICAL USE SMITHKLINE BEECHAM CORPORATION (US) 2005-01-20 WO disclosed