SCHEMBL12824482

SCHEMBL12824482

NCCC(C=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
PNMT P11086 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
ALDH1A1 P00352 2/20 0.37
CDC7 O00311 1/20 0.37
PLK4 O00444 1/20 0.37
CHEK1 O14757 1/20 0.37
DCLK1 O15075 1/20 0.37
MAPK13 O15264 1/20 0.37
PDPK1 O15530 1/20 0.37
DAPK3 O43293 1/20 0.37
DYRK3 O43781 1/20 0.37
ROCK2 O75116 1/20 0.37
RPS6KA5 O75582 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27925692 0.83 SLC6A3 (0.43) SLC6A2SLC6A4SLC6A3ALDH1A1LMNA
SCHEMBL28032633 0.80 SLC6A3 (0.45) SLC6A2SLC6A4SLC6A3ALDH1A1LMNA
SCHEMBL4194753 0.79 SLC6A4 (0.52) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL27257818 0.79 ALDH1A1 (0.40) ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL12825280 0.79 SLC6A2 (0.40) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL19812649 0.78 TAAR1 (0.41) CYP2D6SLC6A2SLC6A4SLC6A3PNMT
SCHEMBL6581676 0.76 SLC6A2 (0.40) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL4680090 0.76 SLC6A2 (0.40) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL12498162 0.76 SLC6A2 (0.48) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6562184 0.73 SLC6A3 (0.39) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295412-A1 Indazole compounds useful as protein kinase inhibitors Vertex Pharmaceuticals Incorporated (US) 2011-03-16 EP disclosed