SCHEMBL12833166

SCHEMBL12833166

C=C(/N=C\C=C/C)n1nc(C(F)(F)F)c(-c2ccc(OC(C)C)c(Cl)c2)c1N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.36
S1PR1 P21453 10/20 0.34
S1PR3 Q99500 1/20 0.34
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMO O15229 2/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRB2 P47870 1/20 0.32
GABRA4 P48169 1/20 0.32
GABRE P78334 1/20 0.32
GABRA6 Q16445 1/20 0.32
GABRG1 Q8N1C3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1006836 0.73 S1PR1 (0.39) S1PR1S1PR3CYP2C9CYP2C19KMO
SCHEMBL16273680 0.56 KMO (0.51) S1PR1S1PR3KMO
SCHEMBL1008749 0.56 POLB (0.43) KMOGABRPGABRDGABRA1GABRB1
SCHEMBL10168911 0.55 CSNK2A1 (0.56) S1PR1S1PR3KMO
SCHEMBL2103199 0.55 CSNK2A1 (0.61) S1PR1S1PR3KMO
SCHEMBL11619472 0.55 RORC (0.40) S1PR1S1PR3CYP2C9CYP2C19KMO
SCHEMBL11619470 0.55 RORC (0.40) S1PR1S1PR3CYP2C9CYP2C19KMO
SCHEMBL11619475 0.55 RORC (0.40) S1PR1S1PR3CYP2C9CYP2C19KMO
SCHEMBL624873 0.55 S1PR1 (0.50) S1PR1S1PR3KMO
SCHEMBL2126187 0.55 S1PR1 (0.50) S1PR1S1PR3KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125789-B1 PYRIMIDINYL PYRAZOLES AS INSECTICIDES AND PARASITICIDE ACTIVE AGENTS BAYER CROPSCIENCE AG (DE) 2011-03-16 EP disclosed