SCHEMBL12835969

SCHEMBL12835969

CCOC(=O)c1cc(C#N)c(N2CC[C@H](N)C2)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.41
P2RY12 Q9H244 7/20 0.40
CHRM2 P08172 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
DRD3 P35462 1/20 0.40
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
PIM1 P11309 1/20 0.39
CLK2 P49760 1/20 0.39
MAP4K2 Q12851 1/20 0.39
CAMK2D Q13557 1/20 0.39
DYRK1A Q13627 1/20 0.39
PIM3 Q86V86 1/20 0.39
AURKB Q96GD4 1/20 0.39
PRKD2 Q9BZL6 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
STK17A Q9UEE5 1/20 0.39
MAP4K5 Q9Y4K4 1/20 0.39
RET P07949 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1514462 0.99 GAA (0.42) GAAP2RY12CHRM2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL1514433 0.99 GAA (0.42) GAAP2RY12CHRM2CYP3A4CYP2C9
SCHEMBL3404525 0.82 ALDH1A1 (0.51) GAAMAPTKDM4EHSD17B10ALDH1A1
SCHEMBL12836341 0.82 P2RY12 (0.41) GAAP2RY12CHRM2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL1514729 0.81 P2RY12 (0.40) GAAP2RY12CHRM2CYP3A4CYP2C9
SCHEMBL1514258 0.81 CTSK (0.47) P2RY12PIM1PIM3RETDPP4
SCHEMBL12835966 0.75 HRH2 (0.44) P2RY12RET
SCHEMBL11441054 0.73 KDM4E (0.51) GAAMAPTKDM4EHSD17B10ALDH1A1
SCHEMBL18430426 0.73 KDM4E (0.47) GAAMAPTKDM4EHSD17B10ALDH1A1
SCHEMBL12895644 0.73 KDM4E (0.45) GAAMAPTKDM4EHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011025799-A1 CATHEPSIN C INHIBITORS GLAXO GROUP LIMITED (GB) 2011-03-03 WO disclosed