SCHEMBL12836611

SCHEMBL12836611

O=C(O)c1cn(C2CC2)c2c(OS(=O)(=O)C(F)(F)F)c(F)ncc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 7/20 0.44
TOP2B Q02880 7/20 0.44
KCNH2 Q12809 6/20 0.42
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 2/20 0.42
HSD17B10 Q99714 2/20 0.42
POLB P06746 2/20 0.42
OPRM1 P35372 2/20 0.42
PRKD3 O94806 1/20 0.42
ALOX15 P16050 1/20 0.42
CLK2 P49760 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
GSK3B P49841 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
OPRD1 P41143 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12835804 0.88 ADRB2 (0.44) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL3397838 0.82 TOP2A (0.55) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL12836323 0.82 TOP2A (0.42) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL12835806 0.79 TOP2A (0.49) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL7841318 0.74 TOP2A (0.55) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL117416 0.72 ADRB2 (0.47) TOP2ATOP2BKCNH2HPGDPOLB
SCHEMBL10412626 0.71 TOP2A (0.47) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL115392 0.71 ADRB2 (0.55) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL7851034 0.71 ALDH1A1 (0.50) TOP2ATOP2BKCNH2ALDH1A1KDM4E
SCHEMBL12836210 0.71 ADRB2 (0.42) TOP2ATOP2BKCNH2HPGDGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011031745-A1 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2011-03-17 WO disclosed