SCHEMBL12836651

SCHEMBL12836651

CCOC(=O)c1cn(C2CC2)c2c3c(c(F)cc2c1=O)N1CCCC1CCOC3

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.49
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
HPGD P15428 3/20 0.43
HSD17B10 Q99714 3/20 0.43
KCNH2 Q12809 6/20 0.42
KMT2A Q03164 2/20 0.41
POLB P06746 2/20 0.41
OPRM1 P35372 2/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
OPRD1 P41143 1/20 0.41
STAT3 P40763 1/20 0.40
PRKD3 O94806 1/20 0.40
ALOX15 P16050 1/20 0.40
CLK2 P49760 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TOP2A P11388 1/20 0.39
TOP2B Q02880 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL116252 0.92 ADRB2 (0.50) ADRB2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL12836931 0.90 ADRB2 (0.48) ADRB2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL115711 0.90 ADRB2 (0.54) ADRB2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL142770 0.90 ADRB2 (0.54) ADRB2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL12836927 0.89 ADRB2 (0.53) ADRB2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL12836938 0.89 ADRB2 (0.47) ADRB2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL12836930 0.87 ADRB2 (0.46) ADRB2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL13625711 0.87 ADRB2 (0.50) ADRB2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL12836652 0.87 ALDH1A1 (0.51) ALDH1A1KDM4EHPGDHSD17B10KCNH2
SCHEMBL116234 0.86 ADRB2 (0.50) ADRB2ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011031743-A1 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2011-03-17 WO disclosed