SCHEMBL12836699

SCHEMBL12836699

Nc1ccc2c(c1)OCCc1cc(Br)sc1-2

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.45
PIK3CA P42336 18/20 0.39
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
PIK3CB P42338 7/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CG P48736 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13655350 0.89 NOTUM (0.45) NOTUMPIK3CAKDM4EGAAMAPT
SCHEMBL988846 0.81 NOTUM (0.62) NOTUMPIK3CAKDM4EGAAMAPT
SCHEMBL1484768 0.80 PIK3CA (0.52) NOTUMPIK3CAPIK3CBPIK3CDPIK3CG
SCHEMBL12836870 0.77 MAP3K14 (0.46) NOTUMPIK3CAKDM4EGAAMAPT
SCHEMBL13655404 0.75 PIK3CA (0.43) NOTUMPIK3CAPIK3CBPIK3CDPIK3CG
SCHEMBL988650 0.73 PIK3CA (0.43) NOTUMPIK3CAPIK3CB
SCHEMBL12535860 0.71 PIK3CA (0.52) NOTUMPIK3CAPIK3CBPIK3CD
SCHEMBL655314 0.70 MAPT (0.52) KDM4EGAAMAPT
SCHEMBL989483 0.70 NOTUM (0.70) NOTUMPIK3CAPIK3CBPIK3CDPIK3CG
SCHEMBL15173260 0.69 NOTUM (0.41) NOTUMPIK3CAMAPTPIK3CBPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011036284-A1 BENZOXEPIN PI3K INHIBITOR COMPOUNDS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2011-03-31 WO disclosed