SCHEMBL12844320

SCHEMBL12844320

CCc1cc(-c2nnc(NC(N)=O)n2-c2cccc3c2ccn3C(C)C)c(O)cc1C

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 14/20 0.37
HSP90AB1 P08238 14/20 0.37
EZH2 Q15910 1/20 0.36
MAP3K5 Q99683 1/20 0.31
P2RX3 P56373 1/20 0.30
P2RX2 Q9UBL9 1/20 0.30
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL444954 0.94 HSP90AA1 (0.39) HSP90AA1HSP90AB1EZH2P2RX3P2RX2
SCHEMBL12287242 0.86 EZH2 (0.33) HSP90AA1HSP90AB1EZH2
SCHEMBL1305321 0.84 EZH2 (0.35) HSP90AA1HSP90AB1EZH2MAP3K5
SCHEMBL421350 0.82 KDM4E (0.35) HSP90AA1HSP90AB1EZH2KDM4EUSP2
SCHEMBL419119 0.80 KDM4E (0.36) HSP90AA1HSP90AB1EZH2KDM4EUSP2
SCHEMBL420062 0.78 KDM4E (0.35) HSP90AA1HSP90AB1EZH2KDM4EUSP2
SCHEMBL12180156 0.77 KDM4E (0.37) HSP90AA1HSP90AB1KDM4EHSD17B10
SCHEMBL1539292 0.75 HSP90AA1 (0.36) HSP90AA1HSP90AB1KDM4ETSHRNPSR1
SCHEMBL12180125 0.74 GOT1 (0.39)
SCHEMBL930906 0.74 SLC9A1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295416-A2 Triazole compounds that modulate HSP90 activity Synta Pharmaceuticals Corp. (US) 2011-03-16 EP disclosed