SCHEMBL12859617

SCHEMBL12859617

c1ccc2c(c1)c1c3c(c4ccccc4c4cccn43)c3c(c4ccccc4c4cccn43)c1n1cccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 5/20 0.39
ATM Q13315 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
CHEK1 O14757 2/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
ALKBH5 Q6P6C2 1/20 0.36
FTO Q9C0B1 1/20 0.36
CYP19A1 P11511 1/20 0.35
POLB P06746 1/20 0.35
ALDH1A1 P00352 3/20 0.35
GAA P10253 2/20 0.35
FABP4 P15090 2/20 0.35
FABP5 Q01469 2/20 0.35
MAPT P10636 2/20 0.35
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25634887 0.82 GPR3 (0.48) GPR3CYP1A2CYP2C19KDM4EATM
SCHEMBL12092119 0.82 GPR3 (0.48) GPR3CYP1A2CYP2C19KDM4EATM
SCHEMBL12270320 0.79 PTPN2 (0.35) KDM4ECHEK1CDK5CDK5R1ALDH1A1
SCHEMBL13089300 0.76
SCHEMBL25634885 0.76 GPR3 (0.42) GPR3CYP1A2CYP2C19KDM4EATM
SCHEMBL12270433 0.76 HPRT1 (0.41) CYP1A2KDM4EATML3MBTL1CHEK1
SCHEMBL12270507 0.76 CHEK1 (0.33) KDM4ECHEK1CDK5CDK5R1ALDH1A1
SCHEMBL19914101 0.74 CYP1A2 (0.47) GPR3CYP1A2CYP2C19KDM4EATM
SCHEMBL25635341 0.71 GPR3 (0.37) GPR3CYP1A2CYP2C19KDM4EATM
SCHEMBL17809837 0.71 KDM4E (0.41) GPR3CYP1A2CYP2C19KDM4EATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110028739-A1 TRI-SUBSTITUTED AROMATIC COMPOUND KEIO UNIVERSITY (JP) 2011-02-03 US disclosed
US-20110028739-A1 TRI-SUBSTITUTED AROMATIC COMPOUND KEIO UNIVERSITY (JP) 2011-02-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110028739-A1 TRI-SUBSTITUTED AROMATIC COMPOUND AHR, AR, ARNT GPR3 20/4885CYP1A2 436/4885CYP2C19 1376/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.