SCHEMBL1286952

SCHEMBL1286952

Nc1nc2[nH]cnc2c(=O)n1-c1cccc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 4/20 0.49
PARP1 P09874 4/20 0.40
TDP1 Q9NUW8 1/20 0.40
GSK3A P49840 2/20 0.37
GSK3B P49841 2/20 0.37
HPGD P15428 2/20 0.37
PI4KA P42356 1/20 0.37
PI4K2B Q8TCG2 1/20 0.37
PI4K2A Q9BTU6 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
CYP2C19 P33261 1/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
POLB P06746 1/20 0.36
PDE4A P27815 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1286937 0.86 GSR (0.37) HCAR1PARP1TDP1HPGDCYP1A2
SCHEMBL1286921 0.85 GSR (0.36) HCAR1PARP1TDP1HPGDCYP1A2
SCHEMBL21768327 0.84 HCAR1 (0.49) HCAR1PARP1GSK3AGSK3BCYP2C19
SCHEMBL637358 0.83 HCAR1 (0.48) HCAR1PARP1ALDH1A1LMNAPDE4A
SCHEMBL8039252 0.81 PARP1 (0.34) HCAR1PARP1GAAKDM4EPOLB
SCHEMBL1286942 0.80 PDE4A (0.45) HCAR1GSK3AGSK3BHPGDGAA
SCHEMBL1286959 0.80 HCAR1 (0.49) HCAR1TDP1GSK3AGSK3BPI4KA
SCHEMBL1286934 0.77 MAPK9 (0.38) HPGDCYP1A2CYP3A4GAACYP2C19
SCHEMBL9283416 0.77 PDE5A (0.46) PARP1CYP2C19KDM4EALDH1A1LMNA
SCHEMBL11610786 0.76 PARP1 (0.42) HCAR1PARP1GSK3AGSK3BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047630-A2 N-ALKYL OR N-ARYL SUBSTITUTED GUANIDE AND BIGUANIDE COMPOUNDS AND METHODS OF THEIR USE TEINTZE MARTIN (US) 2012-04-12 WO disclosed