SCHEMBL1287565

SCHEMBL1287565

CCc1oc2cc(OC)ccc2c1C(=O)c1ccc(OC)cc1

nearest known ligand 0.88

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 10/20 0.88
CYP2C9 P11712 2/20 0.64
CYP3A4 P08684 1/20 0.56
MAPT P10636 1/20 0.56
ALOX15 P16050 1/20 0.56
CNR1 P21554 1/20 0.56
CASP1 P29466 1/20 0.56
CNR2 P34972 1/20 0.56
CASP7 P55210 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
EYA3 Q99504 3/20 0.54
CYP2C19 P33261 4/20 0.54
TTR P02766 2/20 0.53
NR1H4 Q96RI1 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1287454 0.94 SLC22A12 (1.00) SLC22A12CYP2C9CYP3A4MAPTALOX15
SCHEMBL1287515 0.91 SLC22A12 (0.86) SLC22A12CYP2C9MAPTSMN1; SMN2EYA3
SCHEMBL1287600 0.89 SLC22A12 (0.88) SLC22A12CYP2C9MAPTSMN1; SMN2EYA3
SCHEMBL1287462 0.86 CYP2C9 (0.83) SLC22A12CYP2C9CYP3A4MAPTSMN1; SMN2
SCHEMBL14495950 0.86 SLC22A12 (0.70) SLC22A12CYP2C9MAPTCYP2C19
SCHEMBL1287526 0.85 SLC22A12 (1.00) SLC22A12CYP2C9CYP3A4MAPTEYA3
SCHEMBL1287500 0.83 SLC22A12 (0.86) SLC22A12CYP2C9MAPTSMN1; SMN2EYA3
SCHEMBL1287502 0.83 SLC22A12 (1.00) SLC22A12CYP2C9MAPTSMN1; SMN2EYA3
SCHEMBL5241747 0.83 SLC22A12 (0.66) SLC22A12CYP2C9CASP1CASP7CYP2C19
SCHEMBL1287903 0.82 SLC22A12 (0.72) SLC22A12CYP2C9MAPTSMN1; SMN2EYA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10005750-B2 Developing potent urate transporter inhibitors: compounds designed for their uricosuric action J-PHARMA CO., LTD. (JP) 2018-06-26 US disclosed
US-20130225673-A1 DEVELOPING POTENT URATE TRANSPORTER INHIBITORS: COMPOUNDS DESIGNED FOR THEIR URICOSURIC ACTION J-PHARMA CO., LTD. (JP) 2013-08-29 US disclosed
WO-2012048058-A2 DEVELOPING POTENT URATE TRANSPORTER INHIBITORS: COMPOUNDS DESIGNED FOR THEIR URICOSURIC ACTION J-PHARMA CO., LTD. (JP) 2012-04-12 WO disclosed
US-7521570-B2 Medicinal compositions containing 6-hydroxybenzbromarone or salts thereof TORLI PHARMACEUTICAL CO., LTD. (JP) 2009-04-21 US disclosed
US-20070185195-A1 Medicinal compositions containing 6-hydroxybenzbromarone or salts thereof HUMAN CELL SYSTEMS, INC. (JP) 2007-08-09 US disclosed
EP-1767531-A1 MEDICINAL COMPOSITIONS CONTAINING 6-HYDROXYBENZBROMARONE OR SALTS THEREOF Torii Pharmaceutical Co., Ltd. (JP) 2007-03-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10005750-B2 Developing potent urate transporter inhibitors: compounds designed for their uricosuric action SLCO2B1, SLCO2A1, SLC10A6 SLC22A12 19/4885CYP2C9 203/4885CYP3A4 283/4885
US-20130225673-A1 DEVELOPING POTENT URATE TRANSPORTER INHIBITORS: COMPOUNDS DESIGNED FOR THEIR URICOSURIC ACTION SLCO2B1, SLCO2A1, SLC10A6 SLC22A12 19/4885CYP2C9 203/4885CYP3A4 283/4885
US-20070185195-A1 Medicinal compositions containing 6-hydroxybenzbromarone or salts thereof XDH, UGT1A6, SLC10A1 SLC22A12 98/4885CYP2C9 295/4885CYP3A4 441/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.