SCHEMBL1289380

SCHEMBL1289380

NC(CCNC1CC1)c1nc(-c2cc3ccccc3o2)nc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 2/20 0.40
PDE10A Q9Y233 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
VCP P55072 1/20 0.36
SIRT6 Q8N6T7 1/20 0.36
RAB9A P51151 2/20 0.33
SOS1 Q07889 1/20 0.33
KDM4E B2RXH2 2/20 0.33
MPO P05164 1/20 0.33
TACR3 P29371 1/20 0.33
GLA P06280 1/20 0.33
PKM P14618 1/20 0.33
APEX1 P27695 1/20 0.33
RECQL P46063 1/20 0.33
BLM P54132 1/20 0.33
MCL1 Q07820 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 1/20 0.33
ACP1 P24666 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4498518 0.99 MKNK1 (0.39) MKNK1PDE10AADORA2AADORA1VCP
Hydrochloric Acid SCHEMBL4512248 0.85 PDE10A (0.41) MKNK1PDE10ASIRT6RAB9AKDM4E
Hydrochloric Acid SCHEMBL4493037 0.83 PDE10A (0.38) PDE10ASIRT6RAB9AKDM4ETACR3
SCHEMBL1289370 0.73 SIRT6 (0.38) MKNK1PDE10AADORA2AADORA1SIRT6
SCHEMBL12473398 0.71 PDE10A (0.37) MKNK1PDE10AADORA2AADORA1SIRT6
Hydrochloric Acid SCHEMBL4512403 0.71 PDE10A (0.38) MKNK1PDE10ASIRT6RAB9AKDM4E
SCHEMBL12473350 0.70 PDE10A (0.39) MKNK1PDE10ASIRT6RAB9AKDM4E
SCHEMBL12473432 0.69 PDE10A (0.36) MKNK1PDE10AADORA2AADORA1SIRT6
SCHEMBL12473409 0.68 PDE10A (0.35) MKNK1PDE10ASIRT6RAB9AKDM4E
SCHEMBL12473359 0.68 SIRT6 (0.36) MKNK1PDE10ASIRT6RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046207-A1 ANTI-PARASITIC SUBSTITUTED RING FUSED AZINE COMPOUNDS PARACO TECHNOLOGY LIMITED (NZ) 2012-04-12 WO disclosed