SCHEMBL1289765

SCHEMBL1289765

[CH2]C(CC)C(N)=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7852646 0.78
SCHEMBL27292244 0.75
SCHEMBL7860768 0.74
SCHEMBL131555 0.73
SCHEMBL126993 0.73
SCHEMBL1289842 0.73
SCHEMBL28252018 0.71 GPR84 (0.47)
SCHEMBL131933 0.71
SCHEMBL1289796 0.71
SCHEMBL27450897 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 74 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4153133-B1 INJECTABLE PHARMACEUTICAL COMPOSITIONS AND USES THEREOF INTERVET INT BV (NL) 2023-11-08 EP claimed
CN-110327468-A Isoxazoline composition and its purposes in the parasitic infestation for preventing or treating animal 英特维特国际股份有限公司 2019-10-15 CN claimed
CN-108685894-A Soft chewing medicinal product 英特维特国际股份有限公司 2018-10-23 CN claimed
CN-104203214-B soft chewable pharmaceutical product 英特维特国际股份有限公司 2018-05-25 CN claimed
CN-107750159-A Drinking water for sterilization contains vitamin isoxazoline solution 英特维特国际股份有限公司 2018-03-02 CN claimed
CN-106999475-A Use of isoxazoline compounds for the treatment of demodex diseases 英特维特国际股份有限公司 2017-08-01 CN claimed
CN-105992517-A Antiparasitic use of isoxazoline compounds 英特维特国际股份有限公司 2016-10-05 CN claimed
CN-105979944-A Use of isoxazoline derivatives for treating or preventing arthropod infestations in poultry 英特维特国际股份有限公司 2016-09-28 CN claimed
CN-105813651-A Isoxazoline compositions and their use in preventing or treating parasitic infestations of animals 英特维特国际股份有限公司 2016-07-27 CN claimed
CN-105616406-A Topical localized isoxazoline formulation INTERVET INT BV 2016-06-01 CN claimed
CN-104780908-A Manufacture of semi-plastic pharmaceutical dosage units INTERVET INT BV 2015-07-15 CN claimed
CN-104334159-A Solid oral pharmaceutical compositions of isoxazoline compounds INTERVET INT BV 2015-02-04 CN claimed
CN-110327468-A Isoxazoline composition and its purposes in the parasitic infestation for preventing or treating animal 英特维特国际股份有限公司 2019-10-15 CN disclosed
CN-109010296-A The Solid oral pharmaceutical composition of isoxazoline compound 英特维特国际股份有限公司 2018-12-18 CN disclosed
CN-108685894-A Soft chewing medicinal product 英特维特国际股份有限公司 2018-10-23 CN disclosed
CN-108125951-A Local external use's isoxazoline preparation comprising tetraethylene-glycol 英特维特国际股份有限公司 2018-06-08 CN disclosed
EP-0232101-A2 Light-sensitive silver halide color photographic material KONICA CORPORATION (JP) 1987-08-12 EP disclosed
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed