SCHEMBL128991

SCHEMBL128991

[O]Cc1ccc2ccccc2c1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.60
CYP2A6 P11509 1/20 0.60
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
HTR2B P41595 1/20 0.50
MC4R P32245 2/20 0.47
MC5R P33032 2/20 0.47
SIGMAR1 Q99720 1/20 0.47
KMT2A Q03164 1/20 0.47
RAB9A P51151 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
MC3R P41968 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3619110 0.93 CYP1A2 (0.52) CYP1A2CYP2A6HTR2AHTR2CHTR2B
SCHEMBL131160 0.81 CYP1A2 (0.56) CYP1A2CYP2A6HTR2AHTR2CHTR2B
SCHEMBL11719313 0.80 CYP1A2 (0.60) CYP1A2CYP2A6HTR2AHTR2CHTR2B
SCHEMBL29774245 0.80 CYP1A2 (0.60) CYP1A2CYP2A6HTR2AHTR2CHTR2B
SCHEMBL27548336 0.79 ALDH1A1 (0.56) CYP1A2CYP2A6RAB9A
SCHEMBL2838141 0.79 CYP1A2 (0.65) CYP1A2CYP2A6HTR2AHTR2CHTR2B
SCHEMBL6240981 0.79 CYP1A2 (0.65) CYP1A2CYP2A6HTR2AHTR2CHTR2B
SCHEMBL29560700 0.79 CYP1A2 (0.65) CYP1A2CYP2A6HTR2AHTR2CHTR2B
SCHEMBL131604 0.78 CYP1A2 (0.62) CYP1A2CYP2A6MC4RMC5RSIGMAR1
SCHEMBL15352007 0.76 CYP2A6 (0.50) CYP1A2CYP2A6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1438 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116693573-A Column arene bisphosphite ligand, and preparation method and application thereof 北京旭阳科技有限公司 2023-09-05 CN claimed
CN-114460302-A Biological probe and preparation method and application thereof 深圳先进技术研究院 2022-05-10 CN claimed
CN-114441753-A New coronavirus detection test strip and preparation method and application method thereof 深圳先进技术研究院 2022-05-06 CN claimed
CN-114437157-A Sialic acid Neu5Ac derivative and preparation method and application thereof 深圳先进技术研究院 2022-05-06 CN claimed
CN-114181250-A Alkenyl phosphine compound and preparation method thereof 中国石油化工股份有限公司 2022-03-15 CN claimed
CN-106795117-B Heterobicyclic compounds and their use for the treatment of tuberculosis 大塚制药株式会社 2020-06-26 CN claimed
EP-3160977-A2 BIPHENYL AMIDES WITH MODIFIED ETHER GROUPS AS HSP90 INHIBITORS AND HSP70 INDUCERS The University of Kansas (US) 2017-05-03 EP claimed
WO-2015200514-A2 BIPHENYL AMIDES WITH MODIFIED ETHER GROUPS AS HSP90 INHIBITORS AND HSP70 INDUCERS THE UNIVERSITY OF KANSAS (US) 2015-12-30 WO claimed
US-8183383-B2 Protein tyrosine phosphatase 1B inhibitor, preparation methods and uses thereof SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2012-05-22 US claimed
US-RE42164-E1 Hepatitis C inhibitor tri-peptides BOEHRINGER INGELHEIM CANADA LTD. (CA) 2011-02-22 US claimed
EP-0365328-B1 Pyridine derivatives ZENECA LTD (GB) 1996-04-03 EP claimed
US-5495018-A ANTIBIOTIC INTERMEDIATES AMERICAN CYANAMID COMPANY (US) 1996-02-27 US claimed
US-5455271-A Using aromatic amine derivitives as mosquito insecticide THE SCRIPPS RESEARCH INSTITUTE (US) 1995-10-03 US claimed
EP-0582810-A1 Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxyetracyclines as antibiotic agents AMERICAN CYANAMID COMPANY (US) 1994-02-16 EP claimed
WO-1994000420-A1 NOVEL TIGHT-BINDING INHIBITORS OF LEUKOTRIENE A4 HYDROLASE THE SCRIPPS RESEARCH INSTITUTE (US) 1994-01-06 WO claimed
EP-0351282-B1 (1-Hydroxy-2-piperidinyl alkyl)-2-indolone, 2-quinolinones, 2-benzo[b]azepinone, 2-benzimidazolone and 2-quinazolinone derivatives, their preparation and therapeutical use SYNTHELABO (FR) 1993-10-27 EP claimed
US-5053415-A Antiischemic, antiinflammatory, antiarthritic agents, cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-01 US claimed
US-5034401-A Cardiovascular disorders or antiischemia agents SYNTHELABO (FR) 1991-07-23 US claimed
EP-0365328-A2 Pyridine derivatives ZENECA LIMITED (GB) 1990-04-25 EP claimed
EP-0351282-A1 (1-Hydroxy-2-piperidinyl alkyl)-2-indolone, 2-quinolinones, 2-benzo[b]azepinone, 2-benzimidazolone and 2-quinazolinone derivatives, their preparation and therapeutical use SYNTHELABO (FR) 1990-01-17 EP claimed