SCHEMBL12900577

SCHEMBL12900577

Cc1coc(C2CNCCN2)n1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
TACR3 P29371 1/20 0.34
CHRNB2 P17787 1/20 0.32
CHRNA5 P30532 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
PARP1 P09874 1/20 0.32
BMPR1B O00238 2/20 0.31
PDGFRB P09619 2/20 0.31
KDR P35968 2/20 0.31
ACVR1B P36896 2/20 0.31
TGFBR1 P36897 2/20 0.31
TGFBR2 P37173 2/20 0.31
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30
ACVRL1 P37023 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL475667 0.78 CHRM2 (0.44) CHRNB2
SCHEMBL475670 0.78 CHRM2 (0.44) CHRNB2
SCHEMBL2573700 0.73 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3TACR3CHRNB2
SCHEMBL13407530 0.72 HTR2A (0.39) SLC6A2SLC6A4SLC6A3
SCHEMBL12900582 0.71 CHRM2 (0.36) CHRNB2CHRNA5CHRNB4CHRNA3BMPR1B
SCHEMBL6764229 0.70 BMPR1B (0.33) PARP1BMPR1BPDGFRBKDRACVR1B
SCHEMBL30515590 0.69 CYP1A2 (0.32)
SCHEMBL5088449 0.67 CCR1 (0.39) PARP1BMPR1BPDGFRBKDRACVR1B
SCHEMBL12900540 0.67 ROCK2 (0.35) PARP1ROCK2ROCK1
SCHEMBL15046892 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110034469-A1 Heterocyclic Compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-02-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110034469-A1 Heterocyclic Compound BIRC5, XIAP, BIRC2 SLC6A2 401/4885SLC6A4 1305/4885SLC6A3 776/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.