SCHEMBL12903

SCHEMBL12903

CCOC(=O)C(=O)C1CSc2cc(O)ccc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
KDM4E B2RXH2 3/20 0.39
GAA P10253 3/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MEN1 O00255 1/20 0.39
MIF P14174 2/20 0.38
CA12 O43570 3/20 0.36
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA7 P43166 3/20 0.36
CA9 Q16790 3/20 0.36
CA14 Q9ULX7 3/20 0.36
KIF11 P52732 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
PFKFB3 Q16875 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30308393 0.90 KDM4E (0.41) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL24189203 0.90 KDM4E (0.41) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL13212 0.87 MAPT (0.39) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL30308402 0.87 LMNA (0.41) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL25883876 0.87 LMNA (0.41) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL24188767 0.86 KDM4E (0.43) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL30308389 0.86 KDM4E (0.43) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL30460538 0.84 ALDH1A1 (0.41) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL7554 0.84 ALDH1A1 (0.41) ALDH1A1KDM4EGAAMAPTKMT2A
SCHEMBL6985 0.82 POLB (0.37) ALDH1A1KDM4EGAAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058149-A1 TRICYCLIC PYRAZOL AMINE DERIVATIVES MERCK SERONO S.A. (CH) 2011-05-19 WO disclosed