SCHEMBL1292161

SCHEMBL1292161

CCNC(=O)Nc1nc2c[c]cc(/C=N/OC)c2s1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ABL1 P00519 12/20 0.45
PIK3CA P42336 1/20 0.42
PIK3CG P48736 1/20 0.42
PIK3CD O00329 1/20 0.37
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1283010 0.83 ABL1 (0.47) NPC1RAB9ASMN1; SMN2ABL1PIK3CA
SCHEMBL1283009 0.83 ABL1 (0.47) NPC1RAB9ASMN1; SMN2ABL1PIK3CA
SCHEMBL12469564 0.76 NPC1 (0.52) NPC1RAB9ASMN1; SMN2ABL1PIK3CA
SCHEMBL1282508 0.76 ABL1 (0.43) NPC1RAB9ASMN1; SMN2ABL1PIK3CA
SCHEMBL1282511 0.76 ABL1 (0.43) NPC1RAB9ASMN1; SMN2ABL1PIK3CA
SCHEMBL1282587 0.75 ABL1 (0.47) NPC1RAB9ASMN1; SMN2ABL1PIK3CA
SCHEMBL1282583 0.75 ABL1 (0.47) NPC1RAB9ASMN1; SMN2ABL1PIK3CA
SCHEMBL28805227 0.69 NPC1 (0.67) NPC1RAB9ASMN1; SMN2ABL1PIK3CA
SCHEMBL12469595 0.69 NPC1 (0.56) NPC1RAB9ASMN1; SMN2ABL1
SCHEMBL6068145 0.68 NPC1 (0.61) NPC1RAB9ASMN1; SMN2ABL1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2625178-A1 BACTERIA TOPOISOMERASE II INHIBITING 2-ETHYLCARBAMOYLAMINO-1, 3-BENZOTHIAZOL-5-YLS Biota Europe Ltd (GB) 2013-08-14 EP disclosed
WO-2012045124-A1 BACTERIA TOPOISOMERASE II INHIBITING 2-ETHYLCARBAMOYLAMINO-1, 3-BENZOTHIAZOL-5-YLS BIOTA EUROPE LTD (GB) 2012-04-12 WO disclosed