SCHEMBL12949802

SCHEMBL12949802

COc1cccc(C(=O)N[C@@H](C)C(=O)N2CCC[C@H]2C=O)c1C

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PREP P48147 6/20 0.43
FAP Q12884 4/20 0.43
HCRTR1 O43613 1/20 0.42
DRD4 P21917 1/20 0.42
UTS2R Q9UKP6 1/20 0.41
MBOAT4 Q96T53 1/20 0.41
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8288957 0.90 CCR1 (0.44) PREPHCRTR1DRD4UTS2RDRD2
SCHEMBL12949799 0.88 PREP (0.44) PREPFAPHCRTR1DRD4UTS2R
SCHEMBL14181582 0.87 STAT6 (0.42) HCRTR1DRD4UTS2RDRD2
SCHEMBL8286743 0.82 PREP (0.50) PREPFAPHCRTR1DRD4DRD2
SCHEMBL12031331 0.82 CASP1 (0.42) PREPFAPHCRTR1
SCHEMBL16281638 0.81 CNR2 (0.46) PREPFAPHCRTR1DRD4UTS2R
SCHEMBL714622 0.80 NPC1 (0.46) PREP
SCHEMBL12031652 0.80 KMT2A (0.46) UTS2RMBOAT4
SCHEMBL14434719 0.78 ALDH1A1 (0.43)
SCHEMBL6818900 0.78 ALDH1A1 (0.50) PREPFAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2270004-A1 Caspase inhibitors and uses thereof Vertex Pharmceuticals Incorporated (US) 2011-01-05 EP disclosed