SCHEMBL12970525

SCHEMBL12970525

CCOC(=O)c1ccc(-c2cn3cc(F)ccc3n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.54
ALDH1A1 P00352 8/20 0.54
ALDH1A3 P47895 3/20 0.54
CYP11B1 P15538 2/20 0.50
CYP11B2 P19099 2/20 0.50
CLK1 P49759 1/20 0.50
DYRK1A Q13627 1/20 0.50
KDM4E B2RXH2 7/20 0.49
NPC1 O15118 6/20 0.49
RAB9A P51151 6/20 0.49
POLB P06746 2/20 0.49
GAA P10253 2/20 0.49
GLA P06280 1/20 0.49
GABRA2 P47869 1/20 0.49
GABRB2 P47870 1/20 0.49
SMN1; SMN2 Q16637 4/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
MITF O75030 1/20 0.47
KDM5A P29375 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10468516 0.89 NPC1 (0.61) APPALDH1A1ALDH1A3KDM4ENPC1
SCHEMBL12970538 0.85 RAB9A (0.59) APPALDH1A1ALDH1A3CLK1DYRK1A
SCHEMBL12970091 0.85 KDM4E (0.60) ALDH1A1ALDH1A3KDM4ENPC1RAB9A
SCHEMBL3500247 0.83 NPC1 (0.56) ALDH1A1ALDH1A3KDM4ENPC1RAB9A
SCHEMBL2426213 0.82 APP (0.62) APPALDH1A1ALDH1A3CYP11B1CYP11B2
SCHEMBL12970268 0.81 RAB9A (0.63) ALDH1A1ALDH1A3KDM4ENPC1RAB9A
SCHEMBL12970585 0.81 KDM4E (0.65) ALDH1A1KDM4ENPC1RAB9APOLB
SCHEMBL4098270 0.80 KDM4E (0.64) ALDH1A1KDM4ENPC1RAB9APOLB
SCHEMBL21727398 0.79 APP (0.65) APPALDH1A1ALDH1A3CYP11B1CYP11B2
SCHEMBL2128899 0.79 ALDH1A1 (0.72) APPALDH1A1ALDH1A3CLK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012133607-A1 PYRAZOLE COMPOUND アステラス製薬株式会社 (JP) 2012-10-04 WO disclosed