SCHEMBL12993229

SCHEMBL12993229

CNCc1cccc(-c2cccc(OC)c2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.60
PRMT6 Q96LA8 5/20 0.58
CHRM2 P08172 2/20 0.56
CHRM1 P11229 1/20 0.56
CHRM3 P20309 1/20 0.56
EPHX2 P34913 1/20 0.55
CASR P41180 2/20 0.55
MAOB P27338 2/20 0.51
BACE1 P56817 1/20 0.50
ALDH1A1 P00352 2/20 0.49
CYP1A1 P04798 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2E1 P05181 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C8 P10632 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2A6 P11509 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP4B1 P13584 1/20 0.48
CYP2B6 P20813 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29370584 0.89 CHRM2 (0.68) HTR7CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL297410 0.89 CHRM2 (0.68) HTR7CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL10077131 0.88 PRMT6 (0.61) HTR7PRMT6CHRM2CHRM1CHRM3
SCHEMBL24061764 0.83 CHRM2 (0.60) HTR7CHRM2CHRM1CHRM3MAOB
SCHEMBL18015799 0.80 MAOB (0.56) CASRMAOBBACE1CYP1A1CYP1A2
SCHEMBL1252083 0.80 PRMT6 (0.73) HTR7PRMT6EPHX2CYP3A4
SCHEMBL196765 0.79 CYP3A4 (0.73) MAOBALDH1A1CYP1A1CYP1A2CYP2E1
SCHEMBL29489425 0.79 CYP3A4 (0.73) MAOBALDH1A1CYP1A1CYP1A2CYP2E1
SCHEMBL4937029 0.79 FYN (0.56) MAOBBACE1CYP1A1CYP1A2CYP2E1
SCHEMBL7508333 0.79 MAOB (0.54) CHRM2CHRM3CASRMAOBBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2261218-A2 Process for preparing phenyl-, pyridinyl- or pyrimidinyl-substituted imidazoles Eisai R&D Management Co., Ltd. (JP) 2010-12-15 EP disclosed
EP-1757591-A1 CINNAMIDE COMPOUND Eisai R&D Management Co., Ltd. (JP) 2007-02-28 EP disclosed