SCHEMBL13005607

SCHEMBL13005607

CC(C)Cc1cccc(CN(CCN(C)C)Cc2ccc3ccccc3c2)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.56
CALM1 P0DP23 1/20 0.50
CAMKK2 Q96RR4 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
HTR2B P41595 1/20 0.50
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
PYCR1 P32322 1/20 0.42
SIGMAR1 Q99720 2/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005440 0.88 CALM1 (0.59) BCHECALM1CAMKK2HTR2AMEN1
SCHEMBL13061028 0.85 CYP1A2 (0.57) BCHECALM1CAMKK2HTR2AHTR2C
SCHEMBL10039139 0.84 CALM1 (0.62) BCHECALM1CAMKK2HDAC3HDAC1
SCHEMBL13005601 0.84 CYP2D6 (0.46) BCHECALM1CAMKK2HTR2ASIGMAR1
SCHEMBL13005625 0.83 BCHE (0.47) BCHECALM1CAMKK2MEN1KMT2A
SCHEMBL13005681 0.83 CALM1 (0.48) BCHECALM1CAMKK2PYCR1MEN1
SCHEMBL13005722 0.83 CALM1 (0.48) BCHECALM1CAMKK2PYCR1MEN1
SCHEMBL13005707 0.82 CALM1 (0.61) BCHECALM1CAMKK2MEN1KMT2A
SCHEMBL13005718 0.82 CALM1 (0.71) BCHECALM1CAMKK2MEN1KMT2A
SCHEMBL13005546 0.82 CALM1 (0.47) BCHECALM1CAMKK2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed