SCHEMBL13006019

SCHEMBL13006019

Bc1cnc(N)c(O[C@H](C)c2c(Cl)ccc(F)c2Cl)c1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MET P08581 14/20 0.75
JAK2 O60674 2/20 0.66
ALK Q9UM73 4/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14495974 1.00 MET (0.75) METJAK2ALK
SCHEMBL10215004 0.88 MET (0.78) METJAK2ALK
SCHEMBL13005642 0.88 MET (0.78) METJAK2ALK
SCHEMBL5252262 0.88 MET (0.78) METJAK2ALK
SCHEMBL488753 0.86 MET (1.00) METJAK2ALK
SCHEMBL30753168 0.86 MET (1.00) METJAK2ALK
SCHEMBL488503 0.86 MET (0.75) METJAK2ALK
SCHEMBL30753162 0.86 MET (1.00) METJAK2ALK
SCHEMBL29858462 0.86 MET (1.00) METJAK2ALK
SCHEMBL16241930 0.86 MET (1.00) METJAK2ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784396-B1 PYRAZOLE-SUBSTITUTED AMINOHETEROARYL COMPOUNDS AS PROTEIN KINASE INHIBITORS PFIZER (US) 2010-12-22 EP disclosed
WO-2007066185-A2 POLYMORPHS OF A C-MET/HGFR INHIBITOR PFIZER PRODUCTS INC. (US) 2007-06-14 WO disclosed