SCHEMBL13010683

SCHEMBL13010683

Clc1ccnc(-c2nccn2Cc2nc3cccnc3[nH]2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 2/20 0.37
METAP2 P50579 2/20 0.37
METAP1 P53582 2/20 0.37
CCR1 P32246 1/20 0.33
CCR5 P51681 1/20 0.33
CCR8 P51685 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
DRD4 P21917 2/20 0.33
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
GSK3B P49841 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
BRD4 O60885 1/20 0.32
HSD17B10 Q99714 1/20 0.32
KDR P35968 2/20 0.31
KCNH2 Q12809 1/20 0.31
TLR7 Q9NYK1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13010713 0.78 TOP1 (0.40) DRD4BRD4
SCHEMBL13010706 0.77 BRD4 (0.35) DRD4CCNB2CDK1CCNB1GSK3B
SCHEMBL13010459 0.74 DRD4 (0.34) DRD4
SCHEMBL3060393 0.74 LMNA (0.39) LMNA
SCHEMBL13010676 0.73 DRD4 (0.38) DRD4
SCHEMBL13010222 0.73 GRM5 (0.39) METAP2METAP1DRD4CCNB2CDK1
SCHEMBL3062352 0.72 TP53 (0.43) LMNA
SCHEMBL3072577 0.72 TP53 (0.41) LMNA
SCHEMBL3070805 0.72 TP53 (0.36) BRD4LMNAMEN1KMT2A
Acetic Acid SCHEMBL10387126 0.68 METAP2 (0.43) CBFBMETAP2METAP1HSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368342-B3 BENZIMIDAZOLE AND PYRIDYLIMIDAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS NEUROGEN CORP (US) 2010-12-01 EP disclosed