SCHEMBL130221

SCHEMBL130221

[CH2]CCCCC(O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.52
LMNA P02545 1/20 0.50
KDM4E B2RXH2 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
AOC3 Q16853 5/20 0.45
ALDH1A1 P00352 1/20 0.40
BCAT2 O15382 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11234621 0.98 RIPK1 (0.50) RIPK1LMNAKDM4EL3MBTL1AOC3
SCHEMBL6199357 0.93 RIPK1 (0.53) RIPK1LMNAKDM4EL3MBTL1AOC3
SCHEMBL11828179 0.89 RIPK1 (0.61) RIPK1LMNAKDM4EL3MBTL1AOC3
SCHEMBL3591601 0.86 RIPK1 (0.55) RIPK1LMNAKDM4EL3MBTL1AOC3
SCHEMBL7480453 0.86 RIPK1 (0.55) RIPK1LMNAKDM4EL3MBTL1AOC3
SCHEMBL8710104 0.84 RIPK1 (0.61) RIPK1LMNAKDM4EL3MBTL1AOC3
SCHEMBL29860819 0.84 RIPK1 (0.61) RIPK1LMNAKDM4EL3MBTL1AOC3
SCHEMBL4837244 0.84 RIPK1 (0.61) RIPK1LMNAKDM4EL3MBTL1AOC3
SCHEMBL2091869 0.82 HRH1 (0.58)
SCHEMBL3081755 0.81 RIPK1 (0.64) RIPK1LMNAKDM4EL3MBTL1AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426167-B1 Thermally stabilized chlorine containing polymers LAMBERTI SPA (IT) 2013-07-17 EP disclosed
EP-2426167-A1 Thermally stabilized chlorine containing polymers Lamberti SPA (IT) 2012-03-07 EP disclosed
EP-1130017-B1 Azole derivatives and their use as superoxide radical inhibitors OTSUKA PHARMA CO LTD (JP) 2005-06-15 EP disclosed
EP-0934937-B1 Azole derivatives as superoxide radical inhibitor OTSUKA PHARMA CO LTD (JP) 2002-02-27 EP disclosed
US-RE37556-E1 (ALKOXYPHENYL)THIAZOLE DERIVATIVES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-1130017-A2 Azole derivatives and their use as superoxide radical inhibitors OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2001-09-05 EP disclosed
US-6080764-A PROTECTING VARIOUS TISSUE CELLS FROM DISTURBANCES ASSOCIATED WITH ISCHEMIA AND BLOOD REPERFUSION IN HEART, BRAIN, KIDNEY, LUNG AND DIGESTIVE TRACT BY INHIBITING SUPEROXIDE-RELEASE BY NEUTROPHILIC LEUKOCYTES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2000-06-27 US disclosed
EP-0934937-A1 Azole derivatives as superoxide radical inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1999-08-11 EP disclosed
EP-0489869-B1 HYDROXY-ARYL METAL CHELATES FOR DIAGNOSTIC NMR IMAGING GEN HOSPITAL CORP (US) 1998-11-11 EP disclosed
CN-1038586-C Pyrazine derivatives and process for preparing same OTSUKA PHARMA CO LTD (JP) 1998-06-03 CN disclosed
US-5198448-A Cardiovascular disorders OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1993-03-30 US disclosed
CN-1067053-A Pyrazines derivatives and preparation method thereof OTSUKA PHARMA CO LTD (JP) 1992-12-16 CN disclosed
EP-0513387-A1 ACTIVE OXYGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-19 EP disclosed
EP-0511879-A1 Pyrazine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-04 EP disclosed
US-5071856-A CARBOSTYRIL DERIVATIVES AND SALTS THEREOF OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-12-10 US disclosed
US-5053514-A Side effect reduction; carbostyril derivatives OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1991-10-01 US disclosed
CN-1046529-A Carbostyril derivative OTSUKA PHARMA CO LTD (JP) 1990-10-31 CN disclosed
EP-0382185-A2 Carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-08-16 EP disclosed
EP-0355583-A2 Cardiotonics OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed
US-4886809-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-12-12 US disclosed