SCHEMBL13042891

SCHEMBL13042891

C[C@@H](NC(=O)c1cc(N)cc(N(C)S)c1)c1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.58
NPC1 O15118 1/20 0.50
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
BACE1 P56817 15/20 0.48
BACE2 Q9Y5Z0 1/20 0.48
MEN1 O00255 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13042147 0.87 KMT2A (0.60) KMT2ANPC1ALDH1A1LMNABACE1
SCHEMBL13043122 0.86 LMNA (0.51) KMT2ANPC1ALDH1A1LMNABACE1
SCHEMBL13041734 0.86 KMT2A (0.58) KMT2ANPC1ALDH1A1LMNABACE1
SCHEMBL3588334 0.85 BACE1 (0.66) BACE1BACE2
SCHEMBL13042151 0.84 KMT2A (0.54) KMT2ANPC1ALDH1A1LMNABACE1
SCHEMBL13042150 0.83 KMT2A (0.55) KMT2ANPC1ALDH1A1LMNABACE1
SCHEMBL13041735 0.79 KMT2A (0.51) KMT2ANPC1ALDH1A1LMNABACE1
SCHEMBL3594890 0.79 BACE1 (0.64) KMT2ABACE1BACE2
SCHEMBL13041737 0.76 BACE1 (0.52) KMT2ANPC1ALDH1A1LMNABACE1
SCHEMBL12111988 0.75 ALDH1A1 (0.54) KMT2ANPC1ALDH1A1LMNABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7847100-B2 1,3,5-substituted phenyl derivative compounds useful as beta-secretase inhibitors for the treatment of Alzheimer's disease Merck, Sharp & Dohme, Inc. (US) 2010-12-07 US disclosed