SCHEMBL13043392

SCHEMBL13043392

O=C(Nc1ccc2c(c1)CCN2c1c(N2CCC3(CC2)OCCO3)c(=O)c1=O)c1sccc1NCc1ccnc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.48
KIT P10721 3/20 0.48
RAF1 P04049 1/20 0.48
LCK P06239 1/20 0.48
RET P07949 1/20 0.48
CYP3A4 P08684 1/20 0.48
MAP3K20 Q9NYL2 1/20 0.48
RIPK3 Q9Y572 1/20 0.48
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
FLT1 P17948 4/20 0.38
PIN1 Q13526 3/20 0.37
BRAF P15056 2/20 0.35
ALDH1A1 P00352 1/20 0.33
PTPN11 Q06124 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3737666 0.95 KDR (0.48) KDRKITRAF1LCKRET
SCHEMBL13043379 0.91 KDR (0.51) KDRKITRAF1LCKRET
SCHEMBL13043372 0.91 KDR (0.52) KDRKITRAF1LCKRET
SCHEMBL13043393 0.90 KDR (0.52) KDRKITRAF1LCKRET
SCHEMBL13043403 0.90 KDR (0.52) KDRKITRAF1LCKRET
SCHEMBL13043420 0.89 KDR (0.51) KDRKITRAF1LCKRET
SCHEMBL13043389 0.86 KDR (0.54) KDRKITRAF1LCKRET
SCHEMBL3735779 0.86 KDR (0.51) KDRKITRAF1LCKRET
SCHEMBL13043373 0.86 KDR (0.52) KDRKITRAF1LCKRET
SCHEMBL13043410 0.85 KDR (0.47) KDRKITRAF1LCKRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7829717-B2 (Arylamidoaryl)squaramide compounds OSI PHARMACEUTICALS, INC. (US) 2010-11-09 US disclosed
US-7829717-B2 (Arylamidoaryl)squaramide compounds OSI PHARMACEUTICALS, INC. (US) 2010-11-09 US disclosed