SCHEMBL13048293

SCHEMBL13048293

CSc1nnc(-c2ccncc2)n1-c1ccc(O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
TSHR P16473 4/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
HTT P42858 2/20 0.50
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
TP53 P04637 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HSD17B10 Q99714 3/20 0.48
ALOX15 P16050 1/20 0.48
MAPT P10636 1/20 0.46
ALPL P05186 1/20 0.45
ALPG P10696 1/20 0.45
KDM4E B2RXH2 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HDAC3 O15379 1/20 0.44
PTK2 Q05397 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20869674 0.88 HSD17B10 (0.56) ALDH1A1TSHRMEN1KMT2AHTT
SCHEMBL6246142 0.84 ALDH1A1 (0.71) ALDH1A1TSHRMEN1KMT2ATP53
SCHEMBL11919912 0.83 TNKS2 (0.58) ALDH1A1TSHRMEN1KMT2ACYP3A4
SCHEMBL20869595 0.80 TSHR (0.71) ALDH1A1TSHRMEN1KMT2AHTT
SCHEMBL13048294 0.80 HSD17B10 (0.46) ALDH1A1TSHRHTTCYP3A4CYP2C9
SCHEMBL28313035 0.79 MAPK13 (0.53) ALDH1A1TSHRMEN1KMT2AHTT
SCHEMBL11385894 0.78 ALDH1A1 (0.51) ALDH1A1TSHRMEN1KMT2ATP53
SCHEMBL13048284 0.77 HSD17B10 (0.43) ALDH1A1TSHRHTTCYP3A4CYP2C9
SCHEMBL20869724 0.74 PTK2 (0.47) ALDH1A1TSHRMEN1KMT2AHTT
SCHEMBL11068750 0.73 KDM4E (0.49) ALDH1A1TSHRMEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010139966-A1 AZOLE DERIVATIVES AS WTN PATHWAY INHIBITORS OSLO UNIVERSITY HOSPITAL HF (NO) 2010-12-09 WO disclosed