SCHEMBL13060698

SCHEMBL13060698

CCOc1c(C)cccc1-c1cccc(C(=O)NC[C@@H]2CCCN2CC)c1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.53
DRD2 P14416 7/20 0.52
ROCK2 O75116 1/20 0.50
ROCK1 Q13464 1/20 0.50
MCHR2 Q969V1 1/20 0.49
MCHR1 Q99705 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13060827 0.91 ABCG2 (0.53) ABCG2DRD2ROCK2ROCK1KMT2A
SCHEMBL13005479 0.87 ABCG2 (0.49) ABCG2DRD2ROCK2ROCK1MCHR2
SCHEMBL13060816 0.84 ABCG2 (0.62) ABCG2DRD2KMT2A
SCHEMBL13060675 0.84 ABCG2 (0.62) ABCG2DRD2KMT2A
SCHEMBL13060858 0.83 ABCG2 (0.51) ABCG2DRD2ROCK2ROCK1KMT2A
SCHEMBL13005425 0.81 ABCG2 (0.57) ABCG2DRD2ROCK2ROCK1KMT2A
SCHEMBL13006797 0.81 ABCG2 (0.57) ABCG2DRD2ROCK2ROCK1KMT2A
SCHEMBL13005478 0.80 ABCG2 (0.47) ABCG2DRD2ROCK2ROCK1KMT2A
SCHEMBL13060652 0.79 DRD2 (0.60) ABCG2DRD2ROCK2ROCK1KMT2A
SCHEMBL13060677 0.79 DRD2 (0.60) ABCG2DRD2ROCK2ROCK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed