SCHEMBL13060652

SCHEMBL13060652

CCc1cccc(-c2cccc(C(=O)NC[C@H]3CCCN3CC)c2)c1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.60
HTR1A P08908 2/20 0.56
ROCK2 O75116 2/20 0.56
ROCK1 Q13464 2/20 0.56
ABCG2 Q9UNQ0 1/20 0.55
HSD17B10 Q99714 1/20 0.53
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13060677 1.00 DRD2 (0.60) DRD2HTR1AROCK2ROCK1ABCG2
SCHEMBL13005448 0.90 HTR1A (0.53) DRD2HTR1AROCK2ROCK1ABCG2
SCHEMBL13005433 0.90 HTR1A (0.53) DRD2HTR1AROCK2ROCK1ABCG2
SCHEMBL17790224 0.84 ROCK2 (0.61) DRD2HTR1AROCK2ROCK1ABCG2
SCHEMBL18901194 0.83 ROCK2 (0.60) DRD2HTR1AROCK2ROCK1ABCG2
SCHEMBL4572920 0.82 DRD2 (0.60) DRD2HTR1AABCG2HSD17B10KMT2A
SCHEMBL19954197 0.82 ROCK2 (0.59) DRD2HTR1AROCK2ROCK1ABCG2
SCHEMBL11919266 0.82 DRD2 (0.67) DRD2ABCG2HSD17B10
SCHEMBL4341169 0.81 MCHR1 (0.69) DRD2ABCG2HSD17B10KMT2A
SCHEMBL13060816 0.81 ABCG2 (0.62) DRD2ABCG2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed