SCHEMBL13061007

SCHEMBL13061007

CCc1cccc(-c2cccc(C(=O)NCCN3CCCCC3)c2)c1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.64
SMYD2 Q9NRG4 2/20 0.57
CHRM3 P20309 1/20 0.55
APP P05067 1/20 0.55
CACNA1G O43497 4/20 0.53
KMT2A Q03164 2/20 0.53
MEN1 O00255 1/20 0.53
MAP4K4 O95819 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
HPGD P15428 1/20 0.52
PARP1 P09874 1/20 0.52
ATR Q13535 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13060642 0.99 ERN1 (0.62) ERN1SMYD2CHRM3APPCACNA1G
SCHEMBL13060850 0.93 SMYD2 (0.67) ERN1SMYD2CHRM3KMT2AMEN1
SCHEMBL13675357 0.93 PARP1 (0.58) ERN1CACNA1GKMT2AMEN1NPSR1
SCHEMBL12334148 0.92 NPSR1 (0.58) ERN1SMYD2CACNA1GKMT2AMEN1
SCHEMBL13060855 0.91 CHRM3 (0.57) ERN1SMYD2CHRM3CYP2C9PARP1
SCHEMBL13005454 0.88 ERN1 (0.60) ERN1SMYD2APPCACNA1GKMT2A
SCHEMBL13005453 0.86 ERN1 (0.59) ERN1SMYD2APPCACNA1GKMT2A
SCHEMBL5476524 0.86 SMYD2 (0.62) SMYD2KMT2AMEN1HPGDPARP1
SCHEMBL774938 0.84 ERN1 (0.70) ERN1SMYD2APPCACNA1GKMT2A
SCHEMBL13005466 0.81 SMYD2 (0.63) ERN1SMYD2KMT2AMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed