SCHEMBL13070083

SCHEMBL13070083

N=C(Nc1ccc2[nH]cc([C@@H]3CCNC[C@H]3F)c2c1)c1cccs1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 16/20 0.45
NOS1 P29475 16/20 0.45
NMT2 O60551 1/20 0.40
NMT1 P30419 1/20 0.40
HTR2A P28223 1/20 0.39
APP P05067 1/20 0.39
NOS2 P35228 9/20 0.38
SLC6A2 P23975 9/20 0.38
CYP3A4 P08684 5/20 0.38
CYP2D6 P10635 5/20 0.38
KCNH2 Q12809 5/20 0.38
CYP2C19 P33261 4/20 0.38
CYP2C9 P11712 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1122146 0.84 NOS3 (0.61) NOS3NOS1NMT2NMT1APP
SCHEMBL12305072 0.83 NOS3 (0.66) NOS3NOS1APPNOS2
SCHEMBL1122438 0.83 NOS3 (0.66) NOS3NOS1APPNOS2
SCHEMBL13846432 0.79 NOS3 (0.49) NOS3NOS1NOS2SLC6A2CYP3A4
SCHEMBL1122070 0.79 NOS3 (0.65) NOS3NOS1NOS2SLC6A2CYP3A4
SCHEMBL12857201 0.77 NOS3 (0.52) NOS3NOS1NOS2SLC6A2CYP3A4
SCHEMBL13849967 0.76 NOS3 (0.65) NOS3NOS1NOS2SLC6A2CYP3A4
SCHEMBL1122005 0.76 HTR1D (0.64) NOS3NOS1APPNOS2CYP3A4
SCHEMBL13846440 0.76 NOS3 (0.65) NOS3NOS1NOS2SLC6A2CYP3A4
SCHEMBL14507885 0.76 NOS3 (0.42) NOS3NOS1NMT2NMT1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1883451-B1 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON INC (CA) 2010-11-24 EP disclosed