SCHEMBL13070352

SCHEMBL13070352

Cc1[nH]c(C)c(-c2ccc(OCCN3CCC(C(F)(F)F)CC3)nc2)c(=O)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.41
CYP4F2 P78329 1/20 0.39
MCHR1 Q99705 4/20 0.36
TLR7 Q9NYK1 1/20 0.36
KDM1A O60341 2/20 0.35
HRH3 Q9Y5N1 1/20 0.35
ATM Q13315 1/20 0.35
ATR Q13535 1/20 0.35
HTR2A P28223 3/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
PIK3CD O00329 1/20 0.34
PIK3R1 P27986 1/20 0.34
PIK3CG P48736 1/20 0.34
KCNH2 Q12809 3/20 0.34
DRD3 P35462 2/20 0.34
DRD2 P14416 1/20 0.34
CHRM1 P11229 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3394567 0.99 SLC2A1 (0.40) SLC2A1CYP4F2MCHR1TLR7KDM1A
SCHEMBL3394837 0.81 GRIN2B (0.40) SLC2A1KCNH2
SCHEMBL3394476 0.81 JAK3 (0.36) SLC2A1HRH3DRD3DRD2
Hydrochloric Acid SCHEMBL3394572 0.78 DRD3 (0.33) KCNH2DRD3DRD2SIGMAR1
Hydrochloric Acid SCHEMBL3397317 0.77 HRH3 (0.41) MCHR1HRH3KCNH2DRD3DRD2
SCHEMBL13283595 0.74 CYP4F2 (0.37) CYP4F2MCHR1KDM1AHRH3ATM
SCHEMBL4490726 0.72 SLC2A1 (0.61) SLC2A1HDAC6
SCHEMBL3397585 0.72 SLC2A1 (0.43) SLC2A1
SCHEMBL4487955 0.71 SLC2A1 (0.66) SLC2A1HDAC6
SCHEMBL3397533 0.71 SLC2A1 (0.42) SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed