SCHEMBL13075464

SCHEMBL13075464

Bc1c(OC)ncc2[nH]ccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.39
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34
TUBA1A Q71U36 1/20 0.34
TUBA1C Q9BQE3 1/20 0.34
TUBB6 Q9BUF5 1/20 0.34
TUBB2B Q9BVA1 1/20 0.34
TUBB1 Q9H4B7 1/20 0.34
RET P07949 1/20 0.33
TRPA1 O75762 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL113504 0.79 BRD4 (0.39) BRD4MKNK1MKNK2TRPA1MEN1
SCHEMBL9942645 0.72 MKNK1 (0.38) BRD4MKNK1MKNK2CCNKCDK12
SCHEMBL21847766 0.72 MKNK1 (0.38) BRD4MKNK1MKNK2MEN1KMT2A
SCHEMBL29424856 0.69 TRPA1 (0.57) TRPA1DRD1
SCHEMBL21988108 0.69 TRPA1 (0.57) TRPA1DRD1
SCHEMBL113847 0.68 PRKCQ (0.41) TRPA1DRD1
SCHEMBL1473221 0.67 BRD4 (0.40) BRD4MKNK1MKNK2MEN1KMT2A
SCHEMBL27290679 0.67 AXL (0.42) BRD4MKNK1MKNK2CCNKCDK12
SCHEMBL2628910 0.67 AXL (0.42) BRD4MKNK1MKNK2CCNKCDK12
SCHEMBL14329063 0.66 TTBK1 (0.38) BRD4CDK2JAK3TTBK1TTBK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125402-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES NOVARTIS AG (CH) 2010-11-04 WO disclosed