SCHEMBL13075666

SCHEMBL13075666

COc1cc(C=O)c(C2=CCN(C)CC2)c(O)c1C(=O)/C=C/c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 10/20 0.49
MAPT P10636 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
CXCL12 P48061 1/20 0.40
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CDK4 P11802 1/20 0.40
CCNB1 P14635 1/20 0.40
CCND1 P24385 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL746012 0.91 ABCB1 (0.54) ABCB1MAPTNPSR1MAOAMAOB
SCHEMBL13075705 0.91 ABCG2 (0.51) ABCB1MAPTNPSR1MAOAMAOB
SCHEMBL20858996 0.90 ABCB1 (0.51) ABCB1MAPTNPSR1MAOAMAOB
SCHEMBL13075863 0.89 ABCB1 (0.42) ABCB1MAPTNPSR1ABCG2
SCHEMBL7025976 0.88 ABCB1 (0.51) ABCB1MAPTNPSR1MAOAMAOB
SCHEMBL13075834 0.87 NFKB1 (0.47) ABCB1MAPTNPSR1MAOAMAOB
SCHEMBL13075649 0.86 ABCG2 (0.50) MAPTNPSR1MAOAMAOBCCNB2
SCHEMBL3704218 0.83 ABCB1 (0.51) ABCB1MAPTNPSR1ABCG2
SCHEMBL746910 0.82 ABCG2 (0.54) ABCB1MAPTNPSR1MAOBABCG2
SCHEMBL744120 0.82 ABCB1 (0.52) ABCB1MAPTNPSR1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129858-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-11-11 WO disclosed