SCHEMBL13075705

SCHEMBL13075705

COc1cccc(/C=C/C(=O)c2c(OC)cc(C=O)c(C3=CCN(C)CC3)c2O)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.51
ABCB1 P08183 6/20 0.49
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NQO1 P15559 2/20 0.44
MAOB P27338 2/20 0.44
NR1H4 Q96RI1 1/20 0.43
KCNA3 P22001 1/20 0.43
MAPT P10636 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL746910 0.91 ABCG2 (0.54) ABCG2ABCB1CYP1A2CYP3A4CYP2D6
SCHEMBL13075666 0.91 ABCB1 (0.49) ABCG2ABCB1MAOBMAPTNPSR1
SCHEMBL13075863 0.89 ABCB1 (0.42) ABCG2ABCB1MAPTNPSR1
SCHEMBL7028079 0.88 ABCG2 (0.51) ABCG2ABCB1CYP1A2CYP3A4CYP2D6
SCHEMBL13075834 0.88 NFKB1 (0.47) ABCG2ABCB1MAOBKCNA3MAPT
SCHEMBL13075657 0.85 ABCG2 (0.53) ABCG2ABCB1CYP1A2CYP3A4CYP2D6
SCHEMBL13075649 0.84 ABCG2 (0.50) ABCG2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3704218 0.83 ABCB1 (0.51) ABCG2ABCB1MAPTNPSR1
SCHEMBL747096 0.82 MAPT (0.59) ABCB1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL747095 0.82 MAPT (0.59) ABCB1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129858-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-11-11 WO disclosed