SCHEMBL13075889

SCHEMBL13075889

Cc1n[nH]c(C)c1C1=NCCC(C(=O)c2nc3ccc(N4CCCNCC4)nc3[nH]2)=C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
PRKCI P41743 2/20 0.34
HRH4 Q9H3N8 2/20 0.31
HRH3 Q9Y5N1 2/20 0.31
PRKCA P17252 1/20 0.31
PRKCQ Q04759 1/20 0.31
PRKCD Q05655 1/20 0.31
MCHR1 Q99705 1/20 0.31
KLKB1 P03952 1/20 0.31
AURKA O14965 2/20 0.31
RIPK1 Q13546 1/20 0.31
CCNT1 O60563 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CDK9 P50750 1/20 0.31
CDK6 Q00534 1/20 0.31
CDK11A Q9UQ88 1/20 0.31
PARP1 P09874 1/20 0.30
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL111098 0.78 CDK4 (0.40) ROCK2ROCK1PRKCIHRH4HRH3
SCHEMBL113063 0.74 CDK4 (0.42) ROCK2ROCK1AURKACDK4CCND1
SCHEMBL112120 0.67 CDK4 (0.55) HRH4HRH3CDK4CCND1CDK6
SCHEMBL111515 0.67 CDK4 (0.57) HRH3CDK4CCND1CDK6PARP1
SCHEMBL13076251 0.66 CDK4 (0.48) CDK4CCND1CDK6PARP1
SCHEMBL111309 0.65 CDK4 (0.61) CDK4CCND1CDK6PARP1
SCHEMBL2127303 0.64 CDK4 (0.47) HRH3AURKARIPK1CDK4CCND1
SCHEMBL13075590 0.62 PRKCQ (0.37) HRH4HRH3PRKCAPRKCQPRKCD
SCHEMBL111484 0.61 CDK4 (0.62) CDK4CCND1CDK6IRAK4
SCHEMBL5205369 0.60 PRKCA (0.46) HRH4HRH3PRKCAPRKCQPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125402-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES NOVARTIS AG (CH) 2010-11-04 WO disclosed