SCHEMBL13076192

SCHEMBL13076192

C=C(Nc1cc(N2CCC(N(C)C)CC2)ccc1N)C(=O)c1ccc(O)c(-c2cncc3ccccc23)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 5/20 0.46
CDK6 Q00534 5/20 0.46
CCND1 P24385 4/20 0.46
CCND3 P30281 4/20 0.46
CCNA2 P20248 3/20 0.46
CDK2 P24941 3/20 0.46
CCNA1 P78396 3/20 0.46
CDK1 P06493 3/20 0.46
CCNB1 P14635 3/20 0.46
HDAC1 Q13547 1/20 0.37
EGFR P00533 6/20 0.37
ALK Q9UM73 1/20 0.37
CHEK2 O96017 2/20 0.35
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
MMP9 P14780 1/20 0.33
MCHR1 Q99705 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
PLK1 P53350 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL111500 0.75 CDK4 (0.77) CDK4CDK6CCND1CCND3CCNA2
SCHEMBL13076543 0.72 CDK4 (0.64) CDK4CDK6CCND1CCND3CCNA2
SCHEMBL13075596 0.69 EGFR (0.41) EGFRALKPLK1
SCHEMBL23606812 0.68 FGFR4 (0.49) HDAC1EGFR
SCHEMBL112881 0.66 CDK4 (0.74) CDK4CDK6CCND1CCND3CCNA2
SCHEMBL111463 0.66 CDK4 (0.75) CDK4CDK6CCND1CCND3CCNA2
SCHEMBL2142406 0.66 CDK4 (0.78) CDK4CDK6CCND1CCND3CCNA2
SCHEMBL2143680 0.66 CDK4 (0.65) CDK4CDK6CCND1CCND3CCNA2
SCHEMBL111803 0.65 CDK4 (0.80) CDK4CDK6CCND1CCND3CCNA2
SCHEMBL31060547 0.65 CDK4 (0.80) CDK4CDK6CCND1CCND3CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125402-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES NOVARTIS AG (CH) 2010-11-04 WO disclosed