SCHEMBL13093077

SCHEMBL13093077

CNNc1cc(C)nc2c(OCc3c(C)ccnc3C)cccc12

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 19/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12711785 0.80 BDKRB2 (0.62) BDKRB2
SCHEMBL13093085 0.80 BDKRB2 (0.47) BDKRB2
SCHEMBL13093035 0.76 BDKRB2 (0.71) BDKRB2CYP3A4CYP2C19
SCHEMBL13145016 0.76 BDKRB2 (0.71) BDKRB2CYP3A4CYP2C19
SCHEMBL13145018 0.75 BDKRB2 (0.72) BDKRB2
SCHEMBL12711772 0.73 BDKRB2 (0.38) BDKRB2CYP3A4
SCHEMBL13093064 0.71 BDKRB2 (0.56) BDKRB2
SCHEMBL12711756 0.71 BDKRB2 (0.68) BDKRB2
SCHEMBL12711997 0.70 BDKRB2 (0.63) BDKRB2CYP3A4CYP2C19
SCHEMBL12712274 0.69 BDKRB2 (0.46) BDKRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144897-B1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-10-20 EP disclosed
WO-2008116620-A1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2008-10-02 WO disclosed