SCHEMBL13136145

SCHEMBL13136145

Cc1ccnc(Nc2cccc(-c3cnc(C(C)(C)NC(=O)OC(C)(C)C)s3)n2)c1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SYK P43405 13/20 0.48
KARS1 Q15046 6/20 0.48
KDR P35968 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13136148 0.89 KARS1 (0.51) SYKKARS1KDR
SCHEMBL2866531 0.83 SYK (0.47) SYKKARS1KDR
SCHEMBL13135987 0.83 SYK (0.47) SYKKARS1KDR
SCHEMBL13136028 0.82 SYK (0.47) SYKKARS1KDR
SCHEMBL2870010 0.81 SYK (0.49) SYKKARS1KDR
SCHEMBL13136147 0.81 KARS1 (0.55) SYKKARS1KDR
SCHEMBL13136563 0.81 KARS1 (0.48) SYKKARS1KDR
SCHEMBL13136244 0.81 SYK (0.51) SYKKARS1KDR
SCHEMBL13136181 0.80 SYK (0.52) SYKKARS1KDR
SCHEMBL13136180 0.79 SYK (0.47) SYKKARS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7803801-B2 Aminopyridine compounds having Syk inhibitory activity JAPAN TOBACCO, INC. (JP) 2010-09-28 US disclosed
US-7803801-B2 Aminopyridine compounds having Syk inhibitory activity JAPAN TOBACCO, INC. (JP) 2010-09-28 US disclosed